Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates

Siva S. Panda; Abdullah M. Asiri; Mohamed Elagawany; Devan D. Buchanan; Behrad Torkian; Keerthana Bathala; Sean J. Thomas; Jason E. Capito; Muhammad N. Arshad; Abeer N. Al-Romaizan

doi:10.1055/s-0036-1590800

Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates

Siva S. Panda, Abdullah M. Asiri, Mohamed Elagawany, Devan D. Buchanan, Behrad Torkian, Keerthana Bathala, Sean J. Thomas, Jason E. Capito, Muhammad N. Arshad, Abeer N. Al-Romaizan

Research output: Contribution to journal › Article › peer-review

3 Scopus citations

Abstract

Benzotriazole-activated pyrazinoic acid was utilized as a versatile building block for the efficient and convenient synthesis of novel hybrid conjugates of pyrazinoic acid with secondary amines via amino acid linkers in high yields.

Original language	English (US)
Article number	so-2017-d0015-op
Pages (from-to)	50-58
Number of pages	9
Journal	SynOpen
Volume	1
Issue number	1
DOIs	https://doi.org/10.1055/s-0036-1590800
State	Published - Mar 1 2017

Keywords

amino acids
antituberculosis
benzotriazole methodology
pyrazinamide
pyrazinoic acid
secondary amines

ASJC Scopus subject areas

Catalysis
Biomaterials
Materials Science (miscellaneous)
Organic Chemistry

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title = "Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates",

abstract = "Benzotriazole-activated pyrazinoic acid was utilized as a versatile building block for the efficient and convenient synthesis of novel hybrid conjugates of pyrazinoic acid with secondary amines via amino acid linkers in high yields.",

keywords = "amino acids, antituberculosis, benzotriazole methodology, pyrazinamide, pyrazinoic acid, secondary amines",

author = "Panda, {Siva S.} and Asiri, {Abdullah M.} and Mohamed Elagawany and Buchanan, {Devan D.} and Behrad Torkian and Keerthana Bathala and Thomas, {Sean J.} and Capito, {Jason E.} and Arshad, {Muhammad N.} and Al-Romaizan, {Abeer N.}",

note = "Funding Information: We thank the Augusta University and Pamplin Student Research Travel Fund for financial support. Publisher Copyright: Copyright {\textcopyright} 2017 Georg Thieme Verlag Stuttgart · New York.",

year = "2017",

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doi = "10.1055/s-0036-1590800",

language = "English (US)",

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T1 - Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates

AU - Panda, Siva S.

AU - Asiri, Abdullah M.

AU - Elagawany, Mohamed

AU - Buchanan, Devan D.

AU - Torkian, Behrad

AU - Bathala, Keerthana

AU - Thomas, Sean J.

AU - Capito, Jason E.

AU - Arshad, Muhammad N.

AU - Al-Romaizan, Abeer N.

N1 - Funding Information: We thank the Augusta University and Pamplin Student Research Travel Fund for financial support. Publisher Copyright: Copyright © 2017 Georg Thieme Verlag Stuttgart · New York.

PY - 2017/3/1

Y1 - 2017/3/1

N2 - Benzotriazole-activated pyrazinoic acid was utilized as a versatile building block for the efficient and convenient synthesis of novel hybrid conjugates of pyrazinoic acid with secondary amines via amino acid linkers in high yields.

AB - Benzotriazole-activated pyrazinoic acid was utilized as a versatile building block for the efficient and convenient synthesis of novel hybrid conjugates of pyrazinoic acid with secondary amines via amino acid linkers in high yields.

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KW - antituberculosis

KW - benzotriazole methodology

KW - pyrazinamide

KW - pyrazinoic acid

KW - secondary amines

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Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates

Abstract

Keywords

ASJC Scopus subject areas

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