Introduction of histidine units using benzotriazolide activation

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2 Scopus citations


N(α) -Boc-N(im) -(4-toluenesulfonyl-l-histidylbenzotriazole) enables convenient acylation of N-, O-, S-, and C-nucleophiles with no detectable racemization. We report efficient syntheses of novel histidine-containing di-, tri-, and tetra-peptides and models for the preparation of potentially biologically active histidine N-, O-, S-, and C-conjugates.

Original languageEnglish (US)
Pages (from-to)110-7
Number of pages8
JournalJournal of Peptide Science
Issue number2
StatePublished - Feb 2013


  • Histidine
  • Molecular Structure
  • Oligopeptides
  • Tosyl Compounds
  • Triazoles
  • Journal Article
  • Research Support, Non-U.S. Gov't


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