@article{8c74ee41d5ed4b368c2a2308c1db3d60,
title = "Mimicking a proline tripeptide with pyrazolidines and a cyclopentane linker",
abstract = "In this work the five-step assembly of a peptidomimetic structurally resembling Prolyl-Prolyl-Proline tripeptide is reported. Proline units are mimicked by two pyrazolidine rings connected to trans-1,2-cyclopentanedicarboxylic acid. The Pro-Pro-Pro mimetic resembles a tri-l-proline unit but with increased lipophilicity and structural constraints imposed by the linker.",
keywords = "Coupling, Heterocycles, Peptide, Peptidomimetic, Proline",
author = "Peter Vertesaljai and Lebedyeva, {Iryna O.} and Oliferenko, {Alexander A.} and Xin Qi and Junjie Fu and Ostrov, {David A.} and Asiri, {Abdullah M.} and {Dennis Hall}, C. and Alan Katritzky",
note = "Funding Information: We thank the University of Florida and the Kenan Foundation for support with this project. This Letter was also funded in part by generous support from King Abdulaziz University – Saudi Arabia, under grant N o D-006/431 . The authors, therefore, acknowledge the technical and financial support of KAU . The authors are grateful to Mr. Z. Wang for helpful discussion and Dr. M.C.A. Dancel (University of Florida) for HRMS analyses. Publisher Copyright: {\textcopyright} 2015 Elsevier Ltd. All rights reserved. Copyright: Copyright 2016 Elsevier B.V., All rights reserved.",
year = "2015",
month = jul,
day = "13",
doi = "10.1016/j.tetlet.2015.09.063",
language = "English (US)",
volume = "56",
pages = "6653--6655",
journal = "Tetrahedron Letters",
issn = "0040-4039",
publisher = "Elsevier Limited",
number = "48",
}